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Late-stage functionalization

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23 results in Keywords: Late-stage functionalization

Chemistry

Working Paper

Reductive Cleavage of Secondary Sulfonamides: Converting Terminal Functional Groups into Versatile Synthetic Handles

Patrick Fier, Suhong Kim, Kevin M. Maloney

Version 1 posted 03 October 2019

850

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Chemistry

Working Paper

Modular allylation of C(sp3)−H bonds by combining decatungstate photocatalysis and HWE olefination in flow

Luca Capaldo, Stefano Bonciolini, Antonio Pulcinella, Manuel Nuno, Timothy Noel

Version 1 posted 09 November 2021

1,031

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Chemistry

Working Paper

Enantioselective Single and Dual a-C–H Bond Functionalization of Cyclic Amines via Enzymatic Carbene Transfer

Xinkun Ren, Bo M. Couture, Ningyu Liu, Manjinder S. Lall, Jeffrey T. Kohrt, Rudi Fasan

Version 1 posted 17 October 2022

507

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Chemistry

Working Paper

Late-Stage β-C(sp3)–H Deuteration of Carboxylic Acids

Alexander Uttry, Sourjya Mal, Manuel van Gemmeren

Version 2 posted 11 May 2021

813

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Chemistry

Working Paper

Tyrosine Bioconjugation with Hypervalent Iodine

Nina Declas, John R. J. Maynard, Laure Menin, Natalia Gasilova, Sebastian Götze, Jakob L. Sprague, Pierre Stallforth, Stefan Matile, Jerome Waser

Version 1 posted 11 August 2022

563

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Chemistry

Working Paper

Pyridylphosphonium Salts as Alternatives to Cyanopyridines in Radical-Radical Coupling Reactions

Jacob W. Greenwood, Andrew McNally

Version 1 posted 20 January 2021

679

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Chemistry

Working Paper

Sequential C-Selective Difluoromethylation/Pd-Catalyzed Decarboxylative Protonation: An Efficient Access to Tertiary Difluoromethylated Scaffolds

Nicolas Duchemin, Roberto Buccafusca, Marc Daumas, Vincent Ferey, Stellios Arseniyadis

Version 1 posted 08 May 2019

936

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Chemistry

Working Paper

Direct C3-functionalization of indoles with alpha-heteroaryl-substituted methyl alcohols via a metal-free hydrogen autotransfer-type reaction

Ethan Pazur, Nikhil Tasker, Peter Wipf

Version 2 posted 18 October 2023

606

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Chemistry

Working Paper

Metal-Free Click Synthesis of Functional 1-Substituted-1,2,3-Triazoles

Marie-Claire Giel, Christopher J. Smedley, Emily R. R. Mackie, Taijie Guo, Jiajia Dong, Tatiana P. Soares da Costa, John E. Moses

Version 1 posted 15 October 2019

1,035

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Chemistry

Working Paper

Enabling late-stage drug diversification by high-throughput experimentation with geometric deep learning

David F. Nippa, Kenneth Atz, Remo Hohler, Alex T. Müller, Andreas Marx, Christian Bartelmus, Georg Wuitschik, Irene Marzuoli, Vera Jost, Jens Wolfard, Martin Binder, Antonia F. Stepan, David B. Konrad, Uwe Grether, Rainer E. Martin, Gisbert Schneider

Version 2 posted 15 November 2022

2,500

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23 results in Late-stage functionalization in Keywords: Late-stage functionalization

Reductive Cleavage of Secondary Sulfonamides: Converting Terminal Functional Groups into Versatile Synthetic Handles

Modular allylation of C(sp3)−H bonds by combining decatungstate photocatalysis and HWE olefination in flow

Enantioselective Single and Dual a-C–H Bond Functionalization of Cyclic Amines via Enzymatic Carbene Transfer

Late-Stage β-C(sp3)–H Deuteration of Carboxylic Acids

Tyrosine Bioconjugation with Hypervalent Iodine

Pyridylphosphonium Salts as Alternatives to Cyanopyridines in Radical-Radical Coupling Reactions

Sequential C-Selective Difluoromethylation/Pd-Catalyzed Decarboxylative Protonation: An Efficient Access to Tertiary Difluoromethylated Scaffolds

Direct C3-functionalization of indoles with alpha-heteroaryl-substituted methyl alcohols via a metal-free hydrogen autotransfer-type reaction

Metal-Free Click Synthesis of Functional 1-Substituted-1,2,3-Triazoles

Enabling late-stage drug diversification by high-throughput experimentation with geometric deep learning

23 results in Keywords: Late-stage functionalization